CONTRAMOL SR 100MG TAB

About

Contramol SR 100mg Tab, containing tramadol, is a centrally acting opioid analgesic indicated for the management of moderate to moderately severe pain. Its sustained-release (SR) formulation is designed to provide prolonged pain relief over an extended period, typically allowing for less frequent dosing. Tramadol exerts its analgesic effects through a dual mechanism: it acts as a weak agonist at mu-opioid receptors and also inhibits the reuptake of norepinephrine and serotonin, which contributes to its pain-relieving properties by modulating descending pain pathways in the spinal cord.

This medication is particularly useful for chronic pain conditions where consistent pain control is essential to improve a patient's quality of life and functional capacity. The sustained-release mechanism helps to maintain stable plasma concentrations of the drug, reducing fluctuations in pain intensity and minimizing the risk of breakthrough pain. Due to its opioid nature, it requires careful prescribing and monitoring to mitigate risks such as dependence, addiction, and potential side effects, especially in vulnerable populations.

Uses

• Management of moderate to moderately severe chronic pain
• Relief of neuropathic pain (off-label use)
• Post-operative pain management
• Pain associated with musculoskeletal conditions

Directions For Use

Take the tablet whole with water, do not crush, chew, or break it. Can be taken with or without food.

Benefits

• Provides sustained and effective pain relief
• Reduces frequency of dosing due to SR formulation
• Improves overall quality of life for chronic pain sufferers
• Helps manage persistent pain symptoms
• Allows for better sleep and daily functioning
• Dual mechanism of action for comprehensive pain control

Side Effects

• Nausea
• Dizziness
• Constipation
• Headache
• Somnolence
• Vomiting
• Dry mouth
• Sweating
• Itching
• Seizures (rare)
• Respiratory depression (rare)
• Serotonin syndrome (rare)
• Addiction/dependence potential
• Withdrawal symptoms
• Anxiety
• Tremors

Safety Measures

• Alcohol - Avoid alcohol; it significantly increases the risk of central nervous system depression, sedation, and respiratory depression.
• Pregnancy - Not recommended; potential for neonatal opioid withdrawal syndrome and other adverse effects on the fetus.
• Breastfeeding - Not recommended; tramadol passes into breast milk and can cause sedation or respiratory depression in the infant.
• Liver - Use with caution; dose adjustment may be necessary in patients with severe hepatic impairment due to reduced metabolism.
• Kidney - Use with caution; dose adjustment may be necessary in patients with severe renal impairment due to reduced excretion.
• Lung - Use with caution in patients with respiratory conditions (e.g., asthma, COPD) due to the risk of respiratory depression.

Disclaimer

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